An Investigational Study of BG-75202 Alone and in Combination With Other Therapeutic Agents in Adults With Advanced Solid Tumors
Start Date
12/11/2025
Completion Date
1/13/2037
Summary
The purpose of this study is to evaluate the safety, tolerability, pharmacokinetics (PK), pharmacodynamics, and preliminary antitumor activity of BG-75202 (KAT6A/B inhibitor) alone and in combination with other therapies in participants with breast cancer and other advanced solid tumors.
Eligibility Criteria
Age Range: 18 years to No maximum
Interventions
BG-75202
CDK4 Inhibitor
Estrogen Receptor Antagonist
Aromatase Inhibitor
Conditions
Locations
University of Alabama At Birmingham Hospital
Birmingham, Alabama 35294-0004
United States
Yale Cancer Center
New Haven, Connecticut 06510
United States
Washington University in St Louis
St Louis, Missouri 63110-1010
United States
Next Oncology Austin
Austin, Texas 78758
United States
The University of Texas Md Anderson Cancer Center
Houston, Texas 77030-4009
United States
Fred Hutchinson Cancer Research Center
Seattle, Washington 98109-4433
United States
Blacktown Cancer and Haematology Centre
Blacktown, New South Wales NSW 2148
Australia
Chris Obrien Lifehouse
Camperdown, New South Wales NSW 2050
Australia
Cancer Research South Australia
Adelaide, South Australia SA 5000
Australia
Austin Health
Heidelberg, Victoria VIC 3084
Australia
Peter Maccallum Cancer Centre
Melbourne, Victoria VIC 3000
Australia
Cancer Hospital Chinese Academy of Medical Sciences
Beijing, Beijing Municipality 100021
China
Beijing Cancer Hospital
Beijing, Beijing Municipality 100142
China
The First Affiliated Hospital of Xiamen University
Xiamen, Fujian 361003
China
Sun Yat Sen University Cancer Center Huangpu Branch
Guangzhou, Guangdong 510555
China
Harbin Medical University Cancer Hospital
Harbin, Heilongjiang 150000
China
Jiangsu Province Hospital Longjiang Branch
Nanjing, Jiangsu 210036
China
Fudan University Shanghai Cancer Centerpudong
Shanghai, Shanghai Municipality 201321
China
Tianjin Medical University Cancer Institute and Hospital
Tianjin, Tianjin Municipality 300060
China
Sir Run Run Shaw Hospital, Zhejiang University School of Medicine
Hangzhou, Zhejiang 310016
China
Istituto Europeo Di Oncologia
Milan, 20141
Italy
Istituto Nazionale Tumori Fondazione G Pascale
Naples, 80131
Italy
Fondazione Policlinico Universitario Agostino Gemelli
Roma, 00168
Italy
Istituto Clinico Humanitas
Rozzano, 20089
Italy
Hospital Universitario Vall Dhebron
Barcelona, 08035
Spain
Next Oncology Barcelona
Barcelona, 8023
Spain
Hospital Universitario 12 de Octubre
Madrid, 28041
Spain
Hospital Clinico San Carlos
Madrid, 28240
Spain
Hospital Universitario Virgen de La Victoria
Málaga, 29010
Spain